Carbonic anhydrase II in complex with carboxylic acid-based inhibitors
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چکیده
منابع مشابه
Azobenzene-based inhibitors of human carbonic anhydrase II
Aryl sulfonamides are a widely used drug class for the inhibition of carbonic anhydrases. In the context of our program of photochromic pharmacophores we were interested in the exploration of azobenzene-containing sulfonamides to block the catalytic activity of human carbonic anhydrase II (hCAII). Herein, we report the synthesis and in vitro evaluation of a small library of nine photochromic su...
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ژورنال
عنوان ژورنال: Acta Crystallographica Section F Structural Biology Communications
سال: 2019
ISSN: 2053-230X
DOI: 10.1107/s2053230x18018344